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Olanzapine, 5-HT, dopamine, histamine and muscarinic antagonist(AB120736)

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Olanzapine 5 Ht Dopamine Histamine And Muscarinic Antagonist Ab120736  Immunocytochemistry Immunofluorescence Img132884

Olanzapine 5 Ht Dopamine Histamine And Muscarinic Antagonist Ab120736  Chemical Structure Img183728

MW 312.43 g/mol, Purity >99%. 5-HT and D2 antagonist (Ki values are 4 (5-HT2A), 11 (5-HT2C) and 57 (5-HT3), 31 (D1), 11 (D2) and 27 nM (D4)). Additionally, displays activity at: M1, M2, M3, M4, H1, α1 and α2 receptors (Ki are 1.9 at (M1), 18 (M2), 25 (M3), 13 (M4), 19 (α1) and 7 nM (α2)). Atypical antipsychotic. Displays anxiolytic activity.
Specifications
Shipped At Conditions Ambient - Can Ship with Ice
Appropriate Long term Storage Conditions Store at -20°C.
CAS Number 132539-06-1